Product Details
Raloxifene is a chemical compound classified as a selective estrogen receptor modulator (SERM). It is studied in laboratory environments for its interactions with estrogen receptors and associated signaling pathways in experimental models.
The compound is provided strictly for in vitro and non-human research applications, and it is not intended for human use or consumption.
Mechanism of Action
Raloxifene functions as a selective estrogen receptor modulator, interacting with estrogen receptors to influence receptor-mediated signaling pathways. In research systems, it is studied for its ability to bind to receptor subtypes and modulate intracellular signaling cascades associated with transcriptional regulation.
At the molecular level, Raloxifene’s interactions with receptor binding domains are analyzed to understand differential activation or inhibition effects in distinct tissue models. These studies provide insights into receptor-ligand specificity and modulation of downstream molecular pathways.
Chemical Properties of Raloxifene
| Property | Value |
| Compound Name | Raloxifene |
| Classification | Selective Estrogen Receptor Modulator (SERM) |
| Chemical Formula | C28H27NO4S |
| Molecular Weight | 510.05 g/mol |
| CAS Number | 82640-04-8 |
| IUPAC Name | [6-hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl]-[4-(2-piperidin-1-ylethoxy)phenyl]methanone |
| Synonyms | Evista, Keoxifene, LY156758, LY 156758, LY-156758 |
Research Applications
Estrogen Receptor Binding Studies
Raloxifene is applied in experimental systems to examine ligand-receptor interactions and receptor subtype selectivity.
Signaling Pathway Analysis
Research focuses on downstream molecular cascades triggered by receptor binding, including transcriptional modulation and receptor-mediated intracellular pathways.
Differential Modulation Studies
The compound is utilized to explore selective receptor modulation in distinct tissue models, providing mechanistic insights into receptor-ligand specificity.
Why Choose BehemothLabz to Buy Raloxifene for Research
BehemothLabz provides research-grade Raloxifene manufactured under controlled laboratory conditions with strict quality assurance protocols. Each batch undergoes analytical verification to ensure consistency in molecular composition and purity.
Comprehensive documentation, including laboratory testing reports and sourcing transparency, supports reproducibility in experimental settings. BehemothLabz maintains a compliance-focused approach, supplying compounds intended strictly for laboratory-based investigation and analytical research
Disclaimer
Raloxifene is intended strictly for laboratory research and analytical purposes only. It is not intended for use in diagnostic procedures, therapeutic applications, or in vivo studies of any kind.
Any references to biochemical pathways, receptor interactions, or enzymatic processes are provided solely for informational and research-context purposes. This compound must be handled exclusively by qualified professionals in controlled laboratory environments in accordance with applicable regulations and safety guidelines.
Improper handling or use outside of controlled research settings is strictly prohibited.
References
- Hong, S., Chang, J., Jeong, K., & Lee, W. (2021). Raloxifene as a treatment option for viral infections. Journal of microbiology (Seoul, Korea), 59(2), 124–131. https://doi.org/10.1007/s12275-021-0617-7
- Peng, T. R., Lin, H. H., Wang, J. Y., Lee, M. C., & Chen, S. M. (2025). Raloxifene as an Adjuvant Therapy for Patients With Schizophrenia: An Up-To-Date Systematic Review and Meta-Analysis. Brain and behavior, 15(7), e70649. https://doi.org/10.1002/brb3.70649
