Product Details: Deslorelin (Peptide)
Deslorelin is a synthetic analogue of gonadotropin-releasing hormone (GnRH) that exhibits enhanced potency and resistance to enzymatic degradation compared to its endogenous counterpart. Functioning as a GnRH receptor agonist, it binds with high affinity to GnRH receptors located on anterior pituitary cells.
Deslorelin has been investigated for therapeutic potential in various clinical contexts such as hormone-responsive malignancies, endometriosis, and fibroid management.
Mechanism of Action
The pharmacodynamics of Deslorelin involve a two-phase modulation of the hypothalamic-pituitary-gonadal (HPG) axis. Initially, Deslorelin stimulates the anterior pituitary gland, resulting in a transient increase in LH and FSH secretion. This surge promotes follicular maturation, ovulation, and sex hormone production in animal models.
Chemical Properties of Deslorelin (Peptide)
- Molecular Formula: C₆₄H₈₃N₁₇O₁₂
- Molecular Weight: 1282.4 g/mol
- CAS Number: 57773-65-6
- PubChem CID: 5311065
- IUPAC Name: (2S)-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[(2S)-1-[[(2S)-5-(diaminomethylideneamino)-1-[(2S)-2-(ethylcarbamoyl)pyrrolidin-1-yl]-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-5-oxopyrrolidine-2-carboxamide
- Synonyms: Deslorelin, Deslorelina, Desloreline, Somagard
Research Applications of Deslorelin
Deslorelin may examine GnRH receptor activity and signaling behavior in endocrine systems.
This peptide may be applied in models investigating the hypothalamic-pituitary-gonadal axis and its regulatory mechanisms.
Deslorelin is also explored in research involving hormone-related signaling pathways and feedback mechanisms. Findings remain dependent on experimental setup.
Why Buy Deslorelin from BehemothLabz
BehemothLabz keeps product details simple and clear. Each batch is prepared for research use. This helps keep consistency during experiments.
Ordering is direct. Payment is secure. Shipping is available to many locations.This is one option to consider if you require Deslorelin for lab work.
BehemothLabz provides Deslorelin with precise specifications and reliable quality. Every batch is put to the test. Information is easy to understand.We offer 24/7 Customer support and consistent service. Reach out to the support team at support@behemothLabz.com | (307) 429-0990 if you have a question.
Disclaimer: This information is for educational purposes only. We do not allow the human consumption of our products. All products are sold strictly for laboratory and research experiments.
Please review the Terms and Conditions before purchasing. Please research the scientific uses of this product before making any purchases.
Packaging and labeling may differ from what is shown on the website.
References
- Millar, R. P., Lu, Z. L., Pawson, A. J., Flanagan, C. A., Morgan, K., & Maudsley, S. (2004). Gonadotropin-releasing hormone receptors. Endocrine Reviews, 25(2), 235–275.https://pubmed.ncbi.nlm.nih.gov/15082521/
- Conn, P. M., & Crowley, W. F. (1991). Gonadotropin-releasing hormone and its analogs. Annual Review of Medicine, 42, 391–405.https://pubmed.ncbi.nlm.nih.gov/1827224/
- Padula, A. M. (2005). GnRH analogues—agonists and antagonists. Animal Reproduction Science, 88(1–2), 115–126.https://pubmed.ncbi.nlm.nih.gov/16139482/
- PubChem. (n.d.). Deslorelin (CID: 5311065). National Center for Biotechnology Information.https://pubchem.ncbi.nlm.nih.gov/compound/5311065
